2001-1998


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2001

 

Synthesis by chemoselective ligation and biological evaluation of novel cell-permeable PKC-zeta pseudosubstrate lipopeptides
Bonnet, D. ; Thiam, K. ; Loing, E. ; Melnyk, O. ; Gras-Masse, H. J. Med. Chem., 2001, 44, 468-471.
DOI : 10.1021/jm000920s

 

Synthesis of clustered glycoside-antigen conjugates by two one-pot, orthogonal, chemoselective ligation reactions : scope and limitations
Grandjean, C. ; Gras-Masse, H. ; Melnyk, O. Chemistry. A European Journal, 2001, 7, 230-239.
DOI : 10.1002/1521-3765(20010105)7:1<230::AID-CHEM230>3.0.CO;2-L

 

Chemoselective acylation of fully deprotected hydrazino acetyl peptides. Application to the synthesis of lipopeptides
Bonnet, D. ; Ollivier, N. ; Gras-Masse, H. ; Melnyk, O. J. Org. Chem., 2001, 66, 443-449.
DOI : 10.1021/jo0010577

 

Synthesis of an amphiphilic aldehyde using as a key step the condensation of a lipophilic glyoxylic acid amide derivative with tris(hydroxymethyl)aminomethane
Bonnet, D. ; Joly, P. ; Gras-Masse, H. ; Melnyk, O. Tetrahedron Lett., 2001, 42, 1875-1877.

DOI : 10.1016/S0040-4039(01)00032-6

 

A tartric acid-based linker for the solid phase synthesis of C-terminal peptide a-oxo-aldehydes
Melnyk, O. ; Fruchart, J.-S. ; Grandjean, C. ; Gras-Masse, H. J. Org. Chem., 2001, 66, 4153-4160.

DOI : 10.1021/jo001509f

 

Novel hyper-branched designed glycomimetics recognized by the human mannose receptor : Quinic or shikimic acid derivatives as mannose bioisosteres
Grandjean, C. ; Angyalosi, G. ; Loing, E. ; Adriaessens, E. ; Melnyk, O. ; Pancré, V. ; Auriault, C. ; Gras-Masse, H. ChemBiochem, 2001, 2, 747-757.

DOI : 10.1002/1439-7633(20011001)2:10<747::AID-CBIC747>3.0.CO;2-O

 

A novel family of amphilic a-oxo-aldehydes for the site specific modification of peptides by two palmitoyl groups in solution or in liposome suspensions
Bourel-Bonnet, L. ; Gras-Masse, H. ; Melnyk, O. Tetrahedron Letters, 2001, 42, 6851-6853.
DOI : 10.1016/S0040-4039(01)01441-1

 

Methyl phenylacetate enolate generated with P4-tBu Schwesinger base : « naked » or not ?
Fruchart, J.-S. ; Gras-Masse, H. ; Melnyk, O. Tetrahedron Letters, 2001, 42, 9153-9155.

DOI : 10.1016/S0040-4039(01)01994-3

 

2000

 

Chemoselective acylation of hydrazinopeptides : a novel and mild method for the derivatization of peptides with sensitive fatty acids
Bonnet, D. ; Rommens, C. ; Gras-Masse, H. ; Melnyk, O. Tetrahedron Lett., 2000, 41, 45-48.

DOI : 10.1016/S0040-4039(99)02024-9

 

One-pot synthesis of antigens-bearing, lysine-based cluster mannosides using two orthogonal chemoselective ligation reactions
Grandjean, C. ; Rommens, C. ; Gras-Masse, H. ; Melnyk, O. Angew. Chem. Int. Ed., 2000, 39, 1068-1072.

DOI: 10.1002/(SICI)1521-3773(20000317)39:6<1068::AID-ANIE1068>3.0.CO;2-4

 

The deprotection of Lys(Mtt) revisited
Bourel, L. ; Carion, O. ; Gras-Masse, H. ; Melnyk, O. J. Pep. Science, 2000, 6, 264-270.

DOI: 10.1002/1099-1387(200006)6:6<264::AID-PSC248>3.0.CO;2-A

 

Functionalization of peptides and proteins by aldehyde or keto groups
Melnyk, O. ; Fehrentz, J.-A. ; Martinez, J. ; Gras-Masse, H. Biopolymers, 2000, 55, 165-186.

DOI: 10.1002/1097-0282(2000)55:2<165::AID-BIP50>3.0.CO;2-#

 

IL-2Rb agonist P1-30 acts in synergy with IL-2, IL-4, IL-9 and IL-15 : biological and molecular effects
Eckenberg, R. ; Moreau, J.-L. ; Melnyk, O. ; Thèze, J. J. Immunol., 2000, 165, 4312-4314.
DOI: 10.4049/​jimmunol.165.8.4312

 

Structural diversity of human class II histocompatibility molecules induced by peptide ligands
Georges, B. ; Loing, E. ; Neveu, R. ; Melnyk, O. ; Gras-Masse, H. ; Auriault, C. FEBS letters, 2000, 481, 249-254.
DOI : 10.1016/S0014-5793(00)01981-5

 

A novel lipophilic glyoxylic acid derivative for the lipidation of peptides using salt-free hydrazone ligation
Bonnet, D. ; Bourel, L. ; Gras-Masse, H. ; Melnyk, O. Tetrahedron Letters, 2000, 41, 10003-10007.

DOI:10.1016/S0040-4039(00)01784-6

 

1999

 

Chemistry of Hydrazinopeptides : a New Hydroperoxydeamination process
Melnyk, O. ; Rommens, C. ; Gras-Masse, H. Tetrahedron Lett., 1999, 40, 1491-1494.

DOI : 10.1016/S0040-4039(99)00020-9

 

Synthesis of hydrazinopeptides using solid phase N-electrophilic amination. Extention to the Fmoc/tert-butyl strategy and chemistry of the N-N bond in strong acid media
Bonnet, D. ; Samson, F. ; Rommens, C. ; Gras-Masse, H. ; Melnyk, O. J. Peptide Res., 1999, 54, 270-278.

DOI : 10.1034/j.1399-3011.1999.00105.x

 

Reactivity of Lys(NH2) containing peptides towards endopeptidases
Samson, S. ; Bonnet, D. ; Rommens, C. ; Gras-Masse, H. ; Melnyk O. J. Peptide Science, 1999, 5, 352-359.

DOI : 10.1002/(SICI)1099-1387(199908)5:8<352::AID-PSC207>3.0.CO;2-O

 

A new linker for the synthesis of C-terminal peptide a-oxo-aldehydes
Fruchart, J.-S. ; Gras-Masse, H. ; Melnyk, O. Tetrahedron Lett., 1999, 40, 6225-6228.

DOI : 10.1016/S0040-4039(99)01161-2

 

A novel and mild solid phase hydroperoxydeamination reaction
Bonnet, D. ; Rommens, C. ; Gras-Masse, H. ; Melnyk, O. Tetrahedron Lett., 1999, 40, 7315-7318.

DOI : 10.1016/S0040-4039(99)01414-8

 

Convergent synthesis of fluorescein-labelled lysine-based cluster glycosides
Grandjean, C. ; Rommens, C. ; Gras-Masse, H. ; Melnyk, O. Tetrahedron Lett., 1999, 40, 7235-7238.

DOI : 10.1016/S0040-4039(99)01535-X

 

Convergent synthesis of D(-)-quinic and shikimic acid-containing dendrimers as potential C-lectins ligands by thioether ligation of unprotected fragments
Grandjean, C. ; Rommens, C. ; Gras-Masse, H. ; Melnyk, O. J. Chem. Soc. Perkin Trans. I, 1999, 20, 2967-2976.

DOI: 10.1039/a904679h

 

Synthesis, folding and structure of the b-turn mimic modified B1 Domain of Streptococcal Protein G
Odaert, B. ; Jean, F. ; Boutillon, C. ; Buisine, E. ; Melnyk, O. ; Tartar, A. ; Lippens, G. Protein Science, 1999, 8, 2773-2783.

DOI: 10.1110/ps.8.12.2773

 

1998

 

Incorporation of a b-turn mimic in the N-terminal fragment of the B1 domain of streptococcal protein G
Melnyk, O. ; Boutillon, C. ; Draffan, L. ; Odaert, B. ; Jean, F. ; Lippens, G. ; Tartar, A. Letters in Peptide Science, 1998, 5, 147-150.

DOI: 10.1007/BF02443458

 

Synthesis and Structural and Functional Evaluation of a Protein Modified with a b-Turn Mimic
Jean, F. ; Buisine, E. ; Melnyk, O. ; Drobecq, H. ; Odaert, B. ; Hugues, M. ; Lippens, G. ; Tartar, A. J. Am. Chem. Soc., 1998, 120, 6076-6083.
DOI : 10.1021/ja972346o

 

A General Approach to the Synthesis of Polyamine Linked-Monoindolylmaleimides, a New Series of Trypanothione Reductase Inhibitors
Salmon, L. ; Landry, V. ; Melnyk, O. ; Maes, L. ; Sergheraert, C. ; Davioud-Charvet, E. Chem. Pharm. Bull., 1998, 46, 707-710.

DOI: 10.1248/cpb.46.707

 

Identification of a sequence-dependent reversible acylation of tosylarginine in a peptidyl-resin reacted with isonicotinyl p-nitrophenylcarbonate
Melnyk, O. ; Chaurand, P. ; Rommens, C. ; Drobecq, H. ; Wieruszeski, J.-M. ; Spengler, B. ; Gras-Masse, H. J. Peptide Res., 1998, 51, 188-193.

DOI: 10.1111/j.1399-3011.1998.tb01215.x

 

Synthesis of lipopeptides using hydrazone chemical ligation
Melnyk, O. ; Bossus, M. ; David, D. ; Rommens, C. ; Gras-Masse, H. J. Peptide Res., 1998, 52, 180-184.

DOI: 10.1111/j.1399-3011.1998.tb01474.x